Terlipressin

Therapeutic Group

Pituitary And Hypothalamic Hormones And Analogues

Indication Dosage

Bleeding From Oesophageal Varices: 

By IV Inj: 

  • Adult (body weight Up To 50 Kg): Initially 1 Mg, Then 1 Mg Every 4-6 Hours For Up To 72 Hours, To Be Administered Over 1 Minute; 
  • Adult (body weight 50-69 Kg): Initially 1.5 Mg, Then 1 Mg; Every 4-6 Hours For Up To 72 Hours, To Be Administered Over 1 Minute; 
  • Adult (body weight 70 Kg And Above): Initially 2 Mg, Then 1 Mg Every 4-6 Hours For Up To 72 Hours, To Be Administered Over 1 Minute

Content

  • Inj: Terlipressin Acetate 1mg; Powder In Vial And Vial With 5 mlicliluent.

Pregnancy

Avoid Unless Benefits Outweigh Risk

Stability

  • Pituitary & Hypothalamic Hormones & Analogues
  • Vasopressin Analogue

Contra Indications

  • None Known

Precautions

  • None Known

Lactation

  • Caution Advised

Side Effects

  • Abdominal Cramps
  • Arrhythmia
  • Bradycardia
  • Diarrhoea
  • Headache
  • Hypertension
  • Hypotension
  • Pallor
  • Peripheral Ischaemia
  • Angina
  • Bronchospasm
  • Convulsions
  • Hot Flushes
  • Hyponatraemia
  • Intestinal Ischaemia
  • Myocardial Infarction
  • Nausea
  • Pulmonary Oedema
  • Heart Failure
  • Skin Necrosis
  • Respiratory Failure
  • Tachycardia
  • Vomiting.
  • Rare: Dyspnoea
  • Hyperglycaemia
  • Stroke