Tacrolimus

Therapeutic Group

Immunosuppressants

Indication Dosage

Prophylaxis Of Graft Rejection Following Liver Transplantation, Starting 12 Hours After Transplantation: 

  • Adult: Initially 100-200 Mcg/kg Daily In 2 Divided Doses 

Prophylaxis Of Graft Rejection Following Kidney Transplantation, Starting Within 24 Hours Of Transplantation: 

  • Adult: Initially 200-300 Mcg/kg Daily In 2 Divided Doses 

Prophylaxis Of Graft Rejection Following Heart Transplantation Following Antibody Induction, Starting Within 5 Days Of Transplantation: 

  • Adult: Initially 75 Mcg/kg Daily In 2 Divided Doses 

Prophylaxis Of Graft Rejection Following Heart Transplantation Without Antibody Induction, Starting Within 12 Hours Of Transplantation: 

  • Adult: Initially 75 Mcg/kg Daily In 2 Divided Doses 

Allograft Rejection Resistant To Conventional Immunosuppressive Therapy: 

  • Adult: Consult Product Literature Or Seek Specialist Advice

Content

  • Cap 0.5mg /1mg /5mg: Tacrolimus 0.5mg /1mg /5mg.

Pregnancy

Consult with Doctor Or Caution Advised

Stability

  • Calcineurin Inhibitor

Contra Indications

  • Avoid Concurrent Administration With Ciclosporin (care If Patient Has Previously Received Ciclosporin).

Precautions

  • Avoid Concurrent Administration With Ciclosporin (care If Patient Has Previously Received Ciclosporin).

Lactation

  • Consult with Doctor Or Caution Advised

Side Effects

  • Alopecia
  • Anaemia
  • Anorexia
  • Anxiety
  • Arthralgia
  • Ascites
  • Bile-duct Abnormalities
  • Blood Disorders
  • Cholestasis
  • Convulsion
  • Confusion
  • Depression
  • Dizziness
  • Dyspnea
  • Electrolyte Disturbances
  • Gi Disturbance Including Dyspepsia
  • Inflammatory And Ulcerative Disorders
  • Haemorrhage
  • Hepatic Dysfunction
  • Hyperglycaemia
  • Hyperkalaemia
  • Hypertension
  • Hyperuricaemia
  • Hypokalaemia
  • Impaired Hearing
  • Insomnia
  • Ischaemic Events
  • Jaundice
  • Leucopenia
  • Mood Changes
  • Muscle Cramp
  • Oedema
  • Pancytopenia
  • Paraesthesia
  • Parenchymal Lung Disorders
  • Peripheral Neuropathy
  • Photophobia
  • Pleural Effusion
  • Psychosis
  • Renal Failure And Impairment
  • Renal Tubular Necrosis
  • Seizures
  • Sleep Disturbances
  • Sweating
  • Tachycardia
  • Thrombocytopenia
  • Thromboembolic Events
  • Tinnitus
  • Tremor
  • Urinary Abnormalities
  • Visual Disturbances
  • Weight Changes
  • Amnesia
  • Arrhythmia
  • Cardiac Arrest
  • Cardiomyopathy
  • Cataract
  • Cerebrovascular Accident
  • Coagulation Disorders
  • Coma
  • Haemolytic Anaemia
  • Pure Red Cell Aplasia
  • Myasthenia
  • Hirsutism.
  • Rare: Stevens-johnson Syndrome.